API Product portfolio

Axplora, global leader in API supply

Axplora offers a comprehensive portfolio of small molecule APIs. We are a global leader in manufacturing non-sterile and sterile steroids as well as a leading supplier of specialty API products, including 5-ASA, UDCA, High Potent Substances (HPS) and anticancer drugs.

Interested in speaking with one of our experts about your generic drug development needs? Connect with us now!

Table key:

# available for reference 

* non-animal and non-human origin

** submission under preparation

CHE = Chennai, India / CSR = Chasse-sur-Rhône, France / GRO = Gropello, Italy / LEV = Leverkusen, Germany / MRX = Mourenx, France / RAU = Raubling, Germany / VIZ = Vizag, India

Steroids

Active Ingredient
CAS Number
Therapeutic Areas MonographAvailable
Grades
Regulatory
Documentation
Produced in
16α-Hydroxyprednisolone
13951-70-7
Advanced
Intermediate
INTERNAL SPEC.StandardEU DMF
US DMF**
GRO
Amcinonide
51022-69-6
DermatologicUSPMicronizedEU DMFGRO
Beclomethasone
Dipropionate
5534-09-8
RespiratoryPH.EUR.
USP
Standard
Micronized
US DMF#
CEP
SAUDI DMF
CN DMF
GRO
Beclomethasone
Dipropionate
Monohydrate
77011-63-3
RespiratoryPH.EUR.
USP
MicronizedEU DMF
US DMF
GRO
Betamethasone baseAdvanced
Intermediate
PH.EUR.
US DMF
StandardEU DMF
US DMF
GRO
Betamethasone
Dipropionate
5593-20-4
DermatologicPH.EUR.
USP
MicronizedUS DMF#
CEP
SAUDI DMF
GRO
Betamethasone
Valerate
2152-44-5
DermatologicPH.EUR.
USP
MicronizedUS DMF#
JP DMF
CEP
GRO
Brexanolone
516-54-1
CNSINTERNAL SPEC.StandardUS-DMF**GRO
Budesonide
51333-22-3
Respiratory
Gastro-Intestinal
PH.EUR.
USP
JP
MicronizedEU DMF
US DMF#
CEP
JP DMF
SAUDI DMF
GRO
Clascoterone
19608-29-8
DermatologicINTERNAL SPEC.StandardDMF**GRO
Chlormadinone
Acetate
302-22-7
ContraceptivePH.EUR.
JP
MicronizedJP DMF
CEP
GRO
Clobetasol
Propionate
25122-46-7
DermatologicPH.EUR.
USP
MicronizedUS DMF#
JP DMF
CEP
SAUDI DMF
GRO
Clobetasone
Butyrate
25122-57-0
DermatologicPH.EUR.MicronizedEU DMFGRO
Clocortolone
Pivalate
34097-16-0
DermatologicUSPMicronizedEU DMF
US DMF
GRO
Cyproterone
Acetate
427-51-0
Anti-AndrogenPH.EUR.MicronizedUS DMF
CEP
GRO
Delmadinone Acetate
13698-449-2
Anti-Androgen (Veterinary)INTERNAL SPEC.MicronizedEU DMFGRO
Desonide
638-94-8
DermatologicUSPMicronizedEU DMF
US DMF#
CN DMF
GRO
Desonide
Sodium
Phosphate
94087-98-6
OphthalmicINTERNAL
SPEC.
StandardEU DMFGRO
Desoximetasone
382-67-2
Dermatologic
Ophthalmic
USPMicronizedEU DMF
US DMF#
GRO
Dexametasone
50-02-2
Anti-InflammatoryUSPMicronizedEU DMF
US DMF#
GRO
Dexametasone Sodium Phosphate
312-93-6
Anti-InflammatoryPH.Eur.
USP
StandardEU DMFGRO
Diflorasone
Diacetate
2557-49-5

Dermatologic
JP
USP
StandardEU DMFGRO
Diflucortolone
Valerate
59198-70-8
DermatologicBP
JP
MicronizedEU DMF
JP DMF
GRO
Difluprednate
23674-86-4
OphthalmicINTERNAL
SPEC.
MicronizedEU DMF
US DMF#
JP DMF
GRO
Exemestane
107868-30-4
Anti-CancerPH.EUR.
USP
MicronizedUS DMF#
CEP
GRO
Fludrocortisone
Acetate
514-36-3
Adrenocortical
Insufficiency
PH.EUR.
USP
MicronizedUS DMF
CEP
GRO
Fludrocortisone
Base
127-31-1
Anti-InflammatoryINTERNAL
SPEC.
MicronizedEU DMFGRO
Flumethasone
  2135-17-3
Advanced IntermediateINTERNAL
SPEC.
MicronizedEU DMF
US DMF
GRO
Flumethasone
Pivalate
2002-29-1
DermatologicPH.EUR.
USP
MicronizedEU DMFGRO
Flunisolide
Anhydrous
3385-03-3
Anti-AsthmaticUSPMicronizedEU DMF
US DMF#
GRO
Flunisolide
Hemihydrate
77326-96-6
RespiratoryUSPMicronizedEU DMF
US DMF#
GRO
Fluocinonide
356-12-7
DermatologicUSP
BP
MicronizedEU DMF
US DMF#
JP DMF
GRO
Fluocinolone
Acetonide
67-73-2
DermatologicPH.EUR.
USP
MicronizedUS DMF#
JP DMF
CEP
CN DMF
SAUDI DMF
GRO
Fluocortolone hexanoate (Caproate)
303-40-2
DermatologicPH.EUR.MicronizedEU DMFGRO
Fluocortolone pivalate
29205-06-9
DermatologicPH.EUR.MicronizedEU DMFGRO
Fluorometholone
Base
426-13-1
OphthalmicUSP
JP
MicronizedEU DMF
JP DMF
US DMF
GRO
Fluprednidene Acetate
1255-35-2
DermatologicINTERNAL SPEC.StandardEU DMFGRO
Flurandrenolide
1524-88-5
DermatologicUSPMicronizedEU DMF
US DMF#
JP DMF
GRO
Fluticasone
Furoate
397864-44-7
RespiratoryINTERNAL
SPEC.
MicronizedEU DMFGRO
Fluticasone
Propionate
80474-14-2
RespiratoryPH.EUR.
USP
MicronizedUS DMF#
CEP
GRO
Fulvestrant
129453-61-8
Anti-CancerPH.EUR.
USP
StandardUS DMF#
CEP
GRO
Halcinonide
3093-35-4
DermatologicUSPMicronizedEU DMF
US DMF#
CN DMF
GRO
Halometasone
Monohydrate
50629-82-8
DermatologicINTERNAL
SPEC.
MicronizedEU DMFGRO
Hydrocortisone
Acetate
50-03-3
Dermatologic
Ophthalmic
PH.EUR.
USP
MicronizedCEP**GRO
Hydrocortisone hydrogen succinate
2203-97-6
Anti-InflammatoryPH.EUR.
USP
StandardEU DMF
US DMF
GRO
Loteprednol
Etabonate
82034-46-6
OphthalmicINTERNAL
SPEC.
StandardEU DMF
US DMF#
GRO
Medroxyprogesterone
Acetate
71-58-9
ContraceptivePH.EUR.
USP
MicronizedUS DMF
CEP
JP DMF
GRO
Megestrol
Acetate
595-33-5
Anti-CancerPH.EUR.
USP
MicronizedUS DMF#
CEP
GRO
Methylprednisolone Aceponate
86401-95-8
Topical/DermatologicINTERNAL SPEC.Standard
Micronized
EU DMFGRO
Methyltestosterone
58-18-4
Anabolic-
Androgenic
PH.EUR.
USP
MicronizedEU DMF
US DMF#
GRO
Mometasone
Furoate
83919-23-7
Respiratory-
Dermatologic
PH.EUR.
USP
MicronizedUS DMF#
CEP
SAUDI DMF
GRO
Osaterone
Acetate
105149-04-0
Anti-Androgen
(Veterinary)
JPMicronizedEU DMFGRO
Paramethasone
Acetate
1597-82-6
DermatologicINTERNAL
SPEC.
MicronizedEU DMFGRO
Prednisolone
Acetate
52-21-1
DermatologicPH.EUR.
USP
StandardCEPGRO
Prednisolone
Hexanoate (Caproate)
69164-69-8
DermatologicINTERNAL
SPEC.
StandardEU DMFGRO
Prednisolone
Valerate
Acetate
72064-79-0
 
Dermatologic
INTERNAL
SPEC.
MicronizedEU DMF
JP DMF
GRO
Prednisolone
Sodium Metasulfobenzoate
3694-41-5
Anti-InflammatoryINTERNAL
SPEC.
StandardEU DMFGRO
Triamcinolone
124-94-7
Dermatologic
Ophthalmic
PH.EUR.
USP
MicronizedEU DMFGRO
Triamcinolone
Acetonide
76-25-5
Dermatologic
Ophthalmic
PH.EUR.
USP
MicronizedUS DMF#
CEP
GRO
Triamcinolone
Diacetate
67-78-7
Dermatologic
Ophthalmic
USPMicronizedEU DMF
US DMF
GRO
Triamcinolone
Hexacetonide
5611-51-8
Anti-InflammatoryPH.EUR.
USP
Standard
Micronized
US DMF
CEP
GRO

Sterile Steroids

Active Ingredient
CAS Number
Therapeutic Areas MonographAvailable
Grades
Regulatory
Documentation
Produced in
Beclomethasone
Dipropionate
5534-09-8
RespiratoryPH.EUR.
USP
MicronizedEU DMFGRO
Budesonide
51333-22-3
RespiratoryPH.EUR.
USP
MicronizedEU DMF
US DMF
GRO
Hydrocortisone
Acetate
50-03-3
OphthalmicPH.EUR.
USP
MicronizedEU DMFGRO
Loteprednol
Etabonate
82034-46-6
OphthalmicINTERNAL
SPEC.
MicronizedEU DMF
US DMF
GRO
Medroxyprogesterone
Acetate (WHO Pre-Qualified)
71-58-9
ContraceptivePH.EUR.
USP
MicronizedUS DMF#
WHO DMF
GRO
Methylprednisolone
Acetate
53-36-1
Injectable
Anti-Inflammatory
PH.EUR.
USP
MicronizedEU DMF
US DMF#
CEP*
GRO
Prednisolone
Acetate
52-21-1
Ophthalmic
Injectable
Anti-Inflammatory
PH.EUR.
USP
MicronizedUS DMF#
CEP
GRO
Prednisolone
Base
50-24-8
Anti-Inflammatory
(Veterinary)
PH.EUR.
USP
MicronizedEU DMFGRO
Triamcinolone
Acetonide
76-25-5
Injectable
Anti-Inflammatory
PH.EUR.
USP
MicronizedEU DMF
US DMF#
JP DMF
CEP*
GRO

High Potent Substances

Active Ingredient
CAS Number
Therapeutic Areas MonographAvailable
Grades
Regulatory
Documentation
Produced in
Cannabidiol
(CBD, Synthetic)
13956-29-1
VariousDAC (German Drug Codex)StandardEU DMF
US DMF
GRO
Formoterol
Fumarate
Dihydrate
183814-30-4
RespiratoryPH.EUR.
USP
MicronizedUS DMF
CEP
GRO
Tirofiban
Hydrochloride
Monohydrate
150915-40-5
CardiovascularINTERNAL
SPEC.
StandardEU DMF
US DMF
GRO
Salmeterol
Xinafoate
94749-08-3
RespiratoryINTERNAL
SPEC.
MicronizedCEPGRO

Cytotoxics

Active Ingredient
CAS Number
Therapeutic Areas MonographAvailable
Grades
Regulatory
Documentation
Produced in
Busulfan
55-98-1
Anti-CancerPH.EUR.
USP
JP
StandardUS DMF#
CEP
SAUDI DMF
GRO
Melphalan HCl
3223-07-2
Anti-CancerINTERNAL
SPEC.
StandardEU DMF
US DMF#
SAUDI DMF
CN DMF
GRO

Specialty Products

Active Ingredient
CAS Number
Therapeutic Areas MonographAvailable
Grades
Regulatory
Documentation
Produced in
Balsalazide Disodium
150399-21-6
Anti-Inflammatory
Gastrointestinal
USPStandard
Fine
Dense
US DMF#
EU DMF
RAU
CHE
Celecoxib (Form III)
169590-42-5
NSAIDPH.EUR.
USP
Fine
Micronized
CEP
EU DMF
US DMF#
CA DMF
VIZ
Esmolol hydrochloride
81161-17-3
Anti-ArrhythmicAPI QUALITYStandardUS DMF#
CA DMF
EU DMF
CSR
Etoricoxib (Form I)
202409-33-4
ArthritisAPI QUALITYStandard
Micronized
EU DMFVIZ
Indapamide
26807-65-8
Anti-Hypertensive
Diuretic
PH.EUR.Standard
Micronized
CEP
EU DMF
VIZ
L-Cysteine HCL Monohydrate
7048-04-6
VariousPH.EUR.StandardCEP
EU DMF
CHE
L-Cysteine HCl
Anhydrous
52-89-1
VariousAPI QUALITYStandardEU DMFCHE
L-Cystine
56-89-3
VariousPH.EUR.Standard
Fine
CEP
EU DMF
CHE
Magnesium  Orotate
34717-03-8
Dietary SupplementAPI QUALITYStandard
Fine
EU DMFCHE
Mesalamine
Mesalazine
5-Aminosalicylic Acid
ASA
89-57-6
Anti-Inflammatory
Gastrointestinal
PH.EUR.
USP
JP
Dense
Fine
Fine Extra
Coarse
CEP
EU DMF
US DMF#
JP DMF
CA DMF
KR DMF#
TW DMF
BR DMF
CN DMF
TH / ID DMF
RAU
VIZ
Methylene Blue
Methylthioninium Chloride
32680-41-4
Vizualization Agent for Colonoscopies
Methemoglobinemia
PH.EUR.
USP
StandardEU DMF**
US DMF
CEP**
VIZ
6-Methyluracil
626-48-2
Skin Burn Treatment
Dietary Supplement
API QUALITYStandard
Micronized
EU DMF
RU DMF
CHE
N-Acetylcysteine
NAC
616-91-1
Mucolytic
Anti-Oxidant
Parenteral Nutrition
PH.EUR.
USP
Fine
N.A.N.H.*
Pyrogenfree
CEP
EU DMF
US DMF#
CA DMF
BR DMF**
IN REG. CERTIFICATE
RAU
Nitroglycerin
Glyceryl Trinitrate
GTN
55-63-0
Angina
Acute Myocardial Infarction
Severe Hypertension
Acute Coronary Artery Spasms
Pure GTN: INTERNAL SPEC.

Mixtures: Ph. Eur., USP
Pure GTN: DNES

Mixtures: Multiple grades available
Pure GTN:
EU-DMF
US-DMF

Mixtures:
CEP
EU-DMF
US-DMF
JP-DMF
LEV
Omega 3
Eicosapentanoic Acid Ethyl Esther
Icosapent Ethyl
86227-47-6
Anti-Inflammatory
Cardiovascular
API QUALITYStandardUS DMF
CA DMF
EU DMF**
MRX
Propafenone
Hydrochloride
34183-22-7
Anti-ArrhythmicPH.EUR.
USP
Fine
Coarse
Micronized
CEP
EU DMF
US DMF#
CA DMF
KR / CN DMF
BR DMF
TH / ID DMF
RAU
CHE
S-Carboxymethylcysteine
Carbocysteine
SCC
638-23-3
MucolyticPH.EUR.
JP
Standard
Micronized
N.A.N.H.*
CEP
EU DMF
JP DMF
ID DMF
ROW DMF
CHE
S-Carboxymethylcysteine-
L-Lysinate
49673-81-6
MucolyticAPI QUALITYStandard
Dense
N.A.N.H.*
EU DMFCHE
Teriflunomide
163451-81-8
Relapsing Forms Of Multiple SclerosisAPI QUALITYStandardUS DMF
CEP**
VIZ
Ursodeoxycholic Acid
Ursodiol
UDCA
128-13-2
Cholelitholytic AgentPH.EUR.
IP
JP
Standard
Milled
Milled HF
Micronized
CEP
EU DMF
JP DMF
IN REG. CERTIFICATE
BR DMF**
KR DMF
CN DMF**
GRO
Zinc Orotate Dihydrate
60388-02-5
Dietary SupplementAPI QUALITYStandard
Micronized
EU DMFCHE

Developments

Active Ingredient
CAS Number
Therapeutic AreasMonographAvailable
Grades
Regulatory
Documentation
Produced in
Betahistine hydrocholride
5579-84-0
AntivertigoAPI QUALITYUnder DevelopmentDMF
Bile Acid DerivatesPlease contact us if you are looking for such a derivative.   –
Chenodeoxycholic Acid
474-25-9
Cholelithocholic AgentAPI QUALITYUnder DevelopmentDMFVIZ
Cholic Acid
81-25-4
Building Bloc For Bile Acid DerivatesAPI QUALITYUnder DevelopmentDMFVIZ
Estetrol
15183-37-6
ContraceptiveGRO
Isavuconazonium sulfate
946075-13-4
Please contact us if you are looking for such an API.
Lysine Monohydrate
39665-12-8
Please contact us if you are looking for such an API.
Methylprednisolone base
83-43-2
Advanced
Intermediate
PH.EUR.
USP
StandardGRO
Methylprednisolone hydrogen succinate
2921-57-5
Anti-InflammatoryPH.EUR.
USP
StandardGRO
Mometasone
Furoate Monohydrate
141646-00-6
RespiratoryPH.EUR.
USP
MicronizedGRO
Pinaverium BromideFunctional gastrointestinal disordersAPI QUALITYUnder DevelopmentDMF
Segesterone Acetate      
7759-35-5
ContraceptiveGRO
TauroUDCA
14605-22-2
Please contact us if you are looking for such an API.

Interested in speaking with one of our experts about your generic drug development needs? Connect with us now!